09-14-02 05:02
No 356247
What's up folks?! I just found a long forgotten patent on my hardrive, and thought some of you might be interested. The precursors are probably a bitch to make, but the finished product isn't controlled.
Anaesthetic Agents - GB766870
"The present invention is an improvement in or modification of the invention of Application No 34943/53 (Serial No 764,958), and provides a process for the manufacture of anaesthetic agents possessing outstanding properties by building up, according to methods known per se, compounds of the general formula:NH.CO-a O Ikylene-N, C-X (wherein X is a halogen substituent, the naphthalene nucleus may contain further substituents or may be hydrogenated in 54-6-7-8-positions, R is hydrogen, alkyl, aralkyl or cycloalkyl, RI alkyl, aralkyl or cycloalkyl and the alkyl residues, if present, may be linked to each other directly or by means of a hetero atom) and converting these compounds into their salts or quaternary ammonium compounds."
http://l2.espacenet.com/espacenet/viewer
Love my country, fear my government.
(Hive Bee)
09-15-02 02:16
No 356505
Does anybody have comments on quality of product? (how fun is it?)
(PVC-Analog Taste-Tester)
09-15-02 20:58
No 356819
There are a number of patents I have kicking around. I'd be willing to put money into synthing them, but the precursors are hard to find or make.
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US6291499
October 25, 2000
2-Cyclohexyl Benzimidazole NMDA/NR2B Antagonists
Abstract
Novel 4-substituted cyclohexanes substituted in the 1-position with 2-benzimidazoles, 2-imidazopyridines, or 4-imidazoles either directly or through a C.sub.1 -C.sub.4 alkyl, cycloalkyl, hydroxyalkyl, alkoxy or aminoalkyl chain are effective as NMDA NR2B antagonists useful for relieving pain.
U.S. Patent References:
4213994
4695575
4820757
5306723
5436255
5714498
5817756
5889019
4902695
4968678
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Method of manufacture of basic ethers
(stated to have antihistaminic, spasmolytic and anaesthetic properties.)
Patent Number: GB686004
Publication date: 1953-01-14
Applicant: Spofa Spojene Farmaceuticke Zd
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Very frustrating, but...Actually, there is no bright side to that situation. Fuck it, there are plenty of other drugs.
Love my country, fear my government.